Telmisartan-d4
Katalog-Nummer HY-13955S1-5mg
Size : 5mg
Marke : MedChemExpress
Telmisartan-d4 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM[1][2].
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
Telmisartan-d4 Chemische Struktur
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Alle Angiotensin Receptor Isoform-spezifische Produkte anzeigen:
Beschreibung |
Telmisartan-d4 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM[1][2]. |
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In Vitro |
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1]. MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. |
Molekulargewicht |
518.64 |
Formel |
C33H26D4N4O2 |
Unlabeled CAS |
144701-48-4 |
SMILES |
CCCC1=NC2=C(C)C=C(C3=NC4=CC=CC=C4N3C)C=C2N1CC5=C([2H])C([2H])=C(C6=CC=CC=C6C(O)=O)C([2H])=C5[2H] |
Versand | Room temperature in continental US; may vary elsewhere. |
Speicherung |
Please store the product under the recommended conditions in the Certificate of Analysis. |
Reinheit & Dokumentation | |
Verweise |
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Telmisartan-d4 Related Classifications
- Endocrinology Cardiovascular Disease
- Others GPCR/G Protein Autophagy
- Isotope-Labeled Compounds Angiotensin Receptor Autophagy
Molaritätsrechner
Verdünnungsrechner
Die Formel zur Berechnung von Molaritäten
Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
The dilution calculator equation
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Diese Gleichung wird häufig abgekürzt als: C1V1 = C2V2
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Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.
Keywords:
Telmisartan-d4Isotope-Labeled CompoundsAngiotensin ReceptorAutophagyInhibitorinhibitorinhibit